Product Name: CID-2745687
Synonyms: 1-(2,4-difluorophenyl)-5-[[2-[[(1,1-dimethylethyl)amino]thioxomethyl]hydrazinylidene]methyl]-1H-pyrazole-4-carboxylic acid, methyl ester ML-194Medchemexpress
Product Overview: A reversible, competitive antagonist of GPR35, blocking activation by the synthetic agonist pamoic acid with a Ki of 12.8 nM; less potently blocks activation of GPR35 by zaprinast (IC50 = 160 nM); shows ~57-fold selectivity for GPR35 over the related rece
Shipping: wet ice
CAS NO: 1353625-73-6 Presatovir
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C17H19F2N5O2S
SMILES: O=C(OC)C1=C(/C=N/NC(NC(C)(C)C)=S)N(C2=CC=C(F)C=C2F)N=C1Histone Demethylase inhibitors
Molecular Weight: 395.4
Formulation: A crystalline solid
Purity: ≥95%PubMed ID:http://www.bloodjournal.org/content/127/10/1221
